Tamoxifen Citrate 20mg per ml x 30ml
Firstly, Tamoxifen Citrate aka Nolvadex is an antineoplastic nonsteroidal selective estrogen receptor modulator (SERM). Secondly, Tamoxifen Citrate is the trans-isomer of a triphenylethylene derivative chemically.
How Tamoxifen Citrate works:
Tamoxifen competitively inhibits the binding of estradiol to estrogen receptors, therefore preventing the receptor from binding to the estrogen-response element on DNA. As a result, it shows reduction in DNA synthesis and cellular response to estrogen.
In addition, Tamoxifen up-regulates the production of transforming growth factor B (TGFb). Transforming growth factor-β (TGF-β) represents an evolutionarily conserved family of secreted polypeptide factors. For example, they regulate many aspects of physiological embryogenesis and adult tissue homeostasis. The TGF-β family members are also involved in pathophysiological mechanisms that underlie many diseases. Lastly, it down-regulates insulin-like growth factor 1 (IGF 1), a factor that stimulates breast cancer cell growth.
- estrogen receptor antagonist
- a bone density conservation agent
- estrogen receptor modulator
- an angiogenesis inhibitor
- antineoplastic agent
Molecular Formula: C26H29NO
Molecular Mass: 563.62
Chemical name: (Z)2-[4-(1,2-diphenyl-1-butenyl) phenoxy]-N, N-dimethylethanamine 2 hydroxy-1,2,3- propanetricarboxylate (1:1)
THIS PRODUCT IS FOR RESEARCH ONLY
This designation allows the use of research chemicals and peptides strictly for in vitro testing and research, to be handled by qualified and licensed professionals, in laboratory settings only. Bodily introduction or injection of any kind, into humans or animals, is strictly illegal by law.
This product is NOT for human use and can be harmful if ingested. This product is not in a sterile solution. It is not a drug, food, or cosmetic.
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