Exemestane 25mg

Description

Exemestane 25mg per ml x 30ml

Firstly, Exemestane is an aromatase inhibitor (AI) initially developed by Pharmacia & Upjohn for the treatment of female breast cancer patients, specifically post-menopausal patients. Not to mention its use as an adjunct therapy when other first-line treatments for breast cancer (such as Nolvadex) failed.

How Exemestane works:

Because Exemestane is a aromatase inhibitor it possesses the characteristic four ring cycloalkane carbon structure common of all steroidal molecules. The fact that Exemestane is a steroidal aromatase inhibitor is the prime reason as to why it is a suicidal aromatase inhibitor that remains permanently bound to the aromatase enzyme.

For example, as the aromatase enzyme attracts to the steroidal structure of the androgens (Testosterone) it aromatizes into estrogen. Therefore, Exemestane’s chemical structure essentially ‘fools’ the aromatase enzyme into binding with it, only to become inhibited/deactivated. In short, the binding strength is so great, this inhibition becomes permanent for the aromatase enzyme that Exemestane has become bound to.

Possible Benefits:

• lowers estrogen production in the body
• treat certain types of breast cancer (such as hormone-receptor-positive breast cancer) in women after menopause
• helps certain types of breast cancer from returning

Molecular Formula: C₂₀H₂₄O₂

Molecular Mass:       296.4 g/mol

THIS PRODUCT IS FOR RESEARCH ONLY

This designation allows the use of research chemicals and peptides strictly for in vitro testing and research, in laboratory settings only. Bodily introduction or injection of any kind, into humans or animals, is strictly illegal by law. This product is NOT for human use and can be harmful if ingested. This product is not in a sterile solution. It is not a drug, food, or cosmetic.

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